DDR1-IN-1 dihydrochloride
目录号: A21813
DDR1 receptor tyrosine kinase inhibitor
DDR1-IN-1 二盐酸盐是一种强效且选择性的 DDR1 受体酪氨酸激酶抑制剂,其 IC50 为 105 nM;对 DDR2 的抑制效力低 4 倍(IC50 = 413 nM)。
Discription | DDR1-IN-1 dihydrochloride is a potent and selective DDR1 receptor tyrosine kinase inhibitor with an IC50 of 105 nM; 4-fold less potent for DDR2 (IC50 = 413 nM). | ||
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目录号 | A21813 |
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分子式 | C30H33Cl2F3N4O3 |
分子量 | 625.51 |
CAS号 | 1780303-76-5 |
SMILES | CC1=C(C=C(C=C1)NC(C2=CC=C(C(C(F)(F)F)=C2)CN3CCN(CC3)CC)=O)OC4=CC(C5)=C(C=C4)NC5=O.Cl.Cl |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2