DRAK2-IN-1
目录号: A18433
DRAK2 抑制剂
DRAK2-IN-1,化合物16,是一种强效、选择性和与ATP竞争的DRAK2抑制剂,其IC50和Ki值分别为3 nM和0.26 nM。DRAK2-IN-1还对DRAK1具有抑制作用(IC50=51 nM)。
Discription | DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0.26 nM, respectively. DRAK2-IN-1 also has inbitory effect on DRAK1 (IC50=51 nM). |
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目录号 | A18433 |
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分子式 | C21H20N4O3 |
分子量 | 376.41 |
CAS号 | 871837-60-4 |
SMILES | CCCCC(NC1=CC2=C(NC(/C2=C3NC4=C(C=CC=C4)C\3=N\O)=O)C=C1)=O |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2