EI1
目录号: A12711
EZH2 抑制剂
EI1 是一种强效且选择性的小分子抑制剂，针对 EZH2，其半抑制浓度（IC50）值分别为 15 nM（野生型 EZH2）和 13 nM（EZH2 Y641F 突变体）。
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生物活性
| Discription | EI1 is a potent and selective small molecule inhibitor of EZH2 with IC50 values of 15 nM and 13 nM for wild type EZH2 and EZH2 Y641F mutant, respectively. | |||||
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| Cell Research |
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产品信息
| 目录号 | A12711 |
|---|---|
| 分子式 | C23H26N4O2 |
| 分子量 | 390.48 |
| CAS号 | 1418308-27-6 |
| SMILES | CCC(CC)N1C=CC2=C(C=C(C=C21)C#N)C(=O)NCC3=C(C=C(NC3=O)C)C |
| 其他名称 | Ezh2 inhibitor, EI-1, EI 1 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | Warmed: 39 mg/mL (99.87 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 25.61 mL | 128.05 mL | 256.1 mL |
| 0.5 mM | 5.12 mL | 25.61 mL | 51.22 mL |
| 1 mM | 2.56 mL | 12.8 mL | 25.61 mL |
| 5 mM | 0.51 mL | 2.56 mL | 5.12 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 1418308-27-6 | 1418308-27-6 供应商 | 1418308-27-6 花费 | 1418308-27-6 生产商 | 订购 1418308-27-6 | 1418308-27-6 代理商