ELA-21 (human)
目录号: A22977
ELA-21(人类)是一种阿普林受体激动剂,具有 pKi 值为 8.52。ELA-21(人类)完全抑制Forskolin诱导的cAMP产生,并以亚纳摩尔级别的效力刺激β-arrestin的招募。ELA-21(人类)是G蛋白依赖和非依赖途径中的激动剂。
Discription | ELA-21 (human) is an apelin receptor agonist with a pKi of 8.52. ELA-21 (human) completely inhibits Forskolin-induced cAMP production and stimulates β-arrestin recruitment with subnanomolar potencies. ELA-21 (human) is an agonist in G-protein-dependent and -independent pathways. |
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目录号 | A22977 |
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分子式 | C112H184N40O25S3 |
分子量 | 2587.14 |
CAS号 | 2245073-05-4 |
Sequence | Leu-Arg-Lys-His-Asn-Cys-Leu-Gln-Arg-Arg-Cys-Met-Pro-Leu-His-Ser-Arg-Val-Pro-Phe-Pro (Disulfide bridge: Cys6-Cys11) |
Sequence shortening | LRKHNCLQRRCMPLHSRVPFP (Disulfide bridge: Cys6-Cys11) |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2