EMT inhibitor-2
目录号: A18568
EMT 抑制剂
EMT inhibitor-2 抑制由免疫细胞释放的如 IL-1β 和 TGF-β 等物质诱导的上皮-间充质转化(EMT)。EMT inhibitor-2 抑制 CYP3A4 睾酮和 CYP2C9,其 IC50 分别为 49.72 和 5.54 μM。
Discription | EMT inhibitor-2 inhibits epithelial-mesenchymal transition (EMT) induced by substances such as IL-1β and TGF-β released from the immunocytes. EMT inhibitor-2 inhibits CYP3A4 testosteron and CYP2C9 with IC50s of 49.72 and 5.54 μM, respectively. |
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目录号 | A18568 |
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分子式 | C24H26N2O8 |
分子量 | 470.47 |
CAS号 | 2232228-60-1 |
SMILES | COC1=C(O)C2=C(OC(C3=CC=C(OC)C(OC)=C3)=CC2=O)C=C1OCCN(C4)CCNC4=O |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |