ERK1/2 inhibitor 1
目录号: A19596
ERK1/2 抑制剂
ERK1/2 inhibitor 1 是一种高效的、可口服的 ERK1/2 抑制剂,在 1 nM 时显示出 60% 的抑制效果,对 ERK1 和 ERK2 的 IC50 分别为 3.0 nM。
Discription | ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively. | |||||
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Cell Research |
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目录号 | A19596 |
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分子式 | C29H32ClN5O4 |
分子量 | 550.05 |
CAS号 | 2095719-90-5 |
SMILES | ClC1=CN=C(NC2CCOCC2)N=C1C3=CC=C(CN([C@H](C)C(N[C@H](CO)C4=CC=CC(C)=C4)=O)C5=O)C5=C3 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2