ERK5-IN-1
目录号: A16232
ERK5 抑制剂
ERK5-IN-1 显示出对 ERK5 的强效抑制作用,其细胞 EC50 值为 0.19 uM,酶学 IC50 值为 0.087 uM;对 LRRK2[G2019S] 的酶学 IC50 值为 0.026 uM。
Discription | ERK5-IN-1 exhibits potent inhibition of ERK5 with cellular EC50 values of 0.19 uM and enzymatic IC50 values of 0.087 uM and of LRRK2[G2019S] with enzymatic IC50 values of 0.026uM. | |||||
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Targets |
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Cell Research |
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目录号 | A16232 |
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分子式 | C25H29N7O2 |
分子量 | 459.54 |
CAS号 | 1234479-76-5 |
SMILES | O=C1N(C)C2=CN=C(NC3=CC=C(N4CCN(C)CC4)C=C3OC)N=C2N(C)C5=CC=CC=C15 |
其他名称 | ERK5 IN 1, ERK5IN1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2