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Fosaprepitant dimeglumine

Fosaprepitant dimeglumine

Name: Fosaprepitant dimeglumine
SKU: A11069

目录号: A11069

neurokinin-1 receptor 拮抗剂

Fosaprepitant dimeglumine Chemical Structure

CAS NO. 265121-04-8

Fosaprepitant是一种选择性的神经激肽-1（NK-1）受体拮抗剂。

库存：现货

规格	价格	数量
5 mg	￥ 350.00
10 mg	￥ 595.00
25 mg	￥ 1,050.00
10mM * 1mL in DMSO	￥ 1,540.00

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生物活性

Fosaprepitant是一种选择性的神经激肽-1（NK-1）受体拮抗剂。

靶点信息

NK-1 receptor

溶解度 *

In vitro	DMSO	183 mg/mL (182.12 mM)
	Water	123 mg/mL (122.41 mM)
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	9.95 mL	49.76 mL	99.52 mL
0.5 mM	1.99 mL	9.95 mL	19.9 mL
1 mM	1 mL	4.98 mL	9.95 mL
5 mM	0.2 mL	1 mL	1.99 mL

*The above data is based on the productmolecular weight 1004.84. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11069
作用机制	Antagonist (拮抗剂)
M. Wt	1004.84
Formula	C37H56F7N6O16P
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	265121-04-8
Synonyms	MK 0517
SMILES	C[C@H](C1=CC(=CC(=C1)C(F)(F)F)C(F)(F)F)O[C@@H]2[C@@H](N(CCO2)CC3=NC(=O)N(N3)P(=O)(O)O)C4=CC=C(C=C4)F.CNC[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O.CNC[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O