GNE-272
目录号: A12474
CBP/EP300 Inhibitor
GNE-272 是一种针对 CBP/EP300 的溴结构域的强效且选择性的体内探针,其 IC50 值分别为 CBP 0.02 μM、EP300 0.03 μM 和 BRD4 13 μM。
CBP/EP300 Inhibitor
Discription | GNE-272 is a potent and selective in vivo probe for the bromodomains of CBP/EP300 with IC50 values of 0.02, 0.03 and 13 μM for CBP, EP300 and BRD4, respectively. | |||||
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Cell Research |
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目录号 | A12474 |
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分子式 | C22H25FN6O2 |
分子量 | 424.47 |
CAS号 | 1936428-93-1 |
SMILES | CC(N1CCC2=C(C(NC3=C(F)C=C(C4=CN(C)N=C4)C=C3)=NN2[C@@H]5COCC5)C1)=O |
其他名称 | GNE 272, GNE272 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2