GR 159897

Name: GR 159897
SKU: A19862
Price: 2100 CNY
Rating: 5 (288 reviews)

目录号: A19862

NK2 antagonist

GR 159897 是一种高效、选择性、竞争性、能穿透大脑的非肽类拮抗剂，针对缓激肽NK2受体，能够抑制 [3H]GR100679 与 hNK2-CHO 细胞和大鼠结肠膜的结合，其 pKis 分别为 9.51 和 10。该药物能够对抗支气管收缩，并具有类似抗焦虑的活性。

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规格	价格	库存
1mg	¥2,205.00	现货
5mg	¥2,100.00	现货
10mg	¥3,920.00	现货
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Data Sheet

SDS

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生物活性

Discription

GR 159897 is a highly potent, selective, competitive, brain-penetrated non-peptide antagonist at tachykinin NK2 receptors, inhibits binding of [3H]GR100679 to hNK2-CHO cells and rat colon membranes with pKis of 9.51 and 10, respectively. Antagonizes bronchoconstriction, with anxiolytic-like activity.

Targets

Target	Value

产品信息

目录号	A19862
分子式	C23H27FN2O2S
分子量	414.54
CAS号	158848-32-9
SMILES	O=[S@](CC1(OC)CCN(CCC2=CNC3=C2C=C(F)C=C3)CC1)C4=CC=CC=C4
其他名称	GR159897; GR-159897
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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