GR 64349
目录号: A23120
NK2 receptor peptide antagonist
GR 64349 是一种高效且高度选择性的 NK2 受体肽拮抗剂,在大鼠结肠中的 EC50 为 3.7 nM。GR 64349 对 NK1 和 NK3 受体的选择性分别超过 1000 倍和 300 倍。
NK2 receptor peptide antagonist
Discription | GR 64349 is a potent and highly selective NK2 receptor peptide antagonist, with an EC50 of 3.7 nM in rat colon. GR 64349 exhibits selectivity >1000 and >300-fold with respect to NK1 and NK3 receptors, respectively. |
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目录号 | A23120 |
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分子式 | C42H68N10O11S |
分子量 | 921.11 |
CAS号 | 137593-52-3 |
Sequence | Lys-Asp-Ser-Phe-Val-{Aaa}-Leu-Met-NH2 |
Sequence shortening | KDSFV{Aaa}LM-NH2 |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2