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GSK 525762A (I-BET-762)

GSK 525762A (I-BET-762)

Name: GSK 525762A (I-BET-762)
SKU: A11440

目录号: A11440

BET 抑制剂

GSK 525762A (I-BET-762) Chemical Structure

CAS NO. 1260907-17-2

GSK 525762A (I-BET-762)是BET(溴域和末端外)家族的小分子抑制剂。

库存：现货

规格	价格	数量
5 mg	￥ 560.00
10 mg	￥ 840.00
25 mg	￥ 1,680.00
50 mg	￥ 2,520.00
10mM * 1mL in DMSO	￥ 630.00

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产品详情

生物活性

GSK 525762A (I-BET-762)是BET(溴域和末端外)家族的小分子抑制剂。

靶点信息

BET proteins (Cell-free assay)
35 nM

溶解度 *

In vitro	DMSO	72 mg/mL (169.84 mM)
	Water	Insoluble
	Ethanol	Warmed: 36 mg/mL (84.92 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	23.59 mL	117.95 mL	235.9 mL
0.5 mM	4.72 mL	23.59 mL	47.18 mL
1 mM	2.36 mL	11.8 mL	23.59 mL
5 mM	0.47 mL	2.36 mL	4.72 mL

*The above data is based on the productmolecular weight 423.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11440
作用机制	Inhibitor (抑制剂)
M. Wt	423.9
Formula	C22H22ClN5O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1260907-17-2
Synonyms	GSK-525762A, GSK525762A
SMILES	CCNC(=O)C[C@H]1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C