GSK 525768A
目录号: A14134
GSK 525768A 是 GSK 525762A 的对映体化合物,后者是一种强效的小分子抑制剂,能够干扰 BET 家族的溴结构域(Brd2、Brd3 和 Brd4)的功能;GSK 525768A 对 BET 没有活性。
Discription | GSK 525768A is the enantiomer compound of GSK 525762A, which is a potent small molecule inhibitor that disrupt the function of the BET family of bromodomains (Brd2, Brd3, and Brd4); GSK 525768A has NO activity towards BET. |
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目录号 | A14134 |
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分子式 | C22H22ClN5O2 |
分子量 | 423.9 |
CAS号 | 1260530-25-3 |
SMILES | CCNC(=O)C[C@@H]1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C |
其他名称 | GSK525768A, GSK-525768A |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2