GSK1324726A (I-BET726)

Name: GSK1324726A (I-BET726)
SKU: A14133
Price: 245 CNY
Rating: 5 (1 reviews)

目录号: A14133

BET 抑制剂

1 篇发表文献

GSK1324726A（I-BET726）是一种新型、高效、选择性的小分子 BET蛋白 抑制剂，对 BRD2（IC50= 41 nM）、BRD3（IC50= 31 nM）和 BRD4（IC50= 22 nM）具有高亲和力。

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Grouped product items
规格	价格	库存
5mg	¥245.00	现货
10mg	¥455.00	现货
25mg	¥945.00	现货
50mg	¥1,435.00	现货
100mg	¥2,205.00	现货
200mg	¥3,080.00	现货
*10mM 1mL in DMSO**	¥280.00	现货
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重要通知：仅供研究使用。我们不向患者销售。

Data Sheet

SDS

顾客使用 Adooq 产品发表的高质量科研文献

Adooq用户使用GSK1324726A (I-BET726)发表的1篇文献

Zhengjun Liu, .et al. , Cell Death Dis, 2020, May 5;11(5):318 PMID: 32371868

生物活性

Discription

GSK1324726A (I-BET726) is a novel, potent, and selective small molecule inhibitor of BET proteins with high affinity to BRD2 (IC50= 41 nM), BRD3 (IC50= 31 nM), and BRD4 (IC50= 22 nM).

Targets

Target	Value

Cell Research

Cell Line	Type	Value	Description	References

产品信息

目录号	A14133
分子式	C25H23ClN2O3
分子量	434.91
CAS号	1300031-52-0
SMILES	CC1CC(C2=C(N1C(=O)C)C=CC(=C2)C3=CC=C(C=C3)C(=O)O)NC4=CC=C(C=C4)Cl
其他名称	I-BET726, GSK 1324726A, GSK-1324726A, I-BET 726
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro	DMSO	77 mg/mL (177.05 mM)
	Water	Insoluble
	Ethanol	77 mg/mL (177.05 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	22.99 mL	114.97 mL	229.93 mL
0.5 mM	4.6 mL	22.99 mL	45.99 mL
1 mM	2.3 mL	11.5 mL	22.99 mL
5 mM	0.46 mL	2.3 mL	4.6 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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