GSK2801

Name: GSK2801
SKU: A14015

目录号: A14015

BAZ2A and BAZ2B 抑制剂

GSK2801 Chemical Structure

CAS NO. 1619994-68-1

GSK2801是BAZ2家族含溴结构域蛋白的强效抑制剂。

库存：现货

规格	价格	数量
10 mg	￥ 490.00
25 mg	￥ 980.00
50 mg	￥ 1,540.00

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生物活性

GSK2801是BAZ2家族含溴结构域蛋白的强效抑制剂。

靶点信息

BAZ2B	BAZ2A
136 nM(Kd)	257 nM(Kd)

溶解度 *

In vitro (25°C)	DMSO	Warmed: 67 mg/mL (180.37 mM)
	Water	Insoluble
	Ethanol	Warmed: 6 mg/mL (16.15 mM)
In vivo	0.5% CMC+1% Tween 80	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	26.92 mL	134.58 mL	269.15 mL
0.5 mM	5.38 mL	26.92 mL	53.83 mL
1 mM	2.69 mL	13.46 mL	26.92 mL
5 mM	0.54 mL	2.69 mL	5.38 mL

*The above data is based on the productmolecular weight 371.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A14015
作用机制	Inhibitor (抑制剂)
M. Wt	371.54
Formula	C20H21NO4S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1619994-68-1
Synonyms	GSK-2801, GSK 2801
SMILES	CCCOC1=CC2=C(C=C(N2C=C1)C(=O)C)C3=CC=CC=C3S(=O)(=O)C