GSK3004774
目录号: A19779
CaSR 激动剂
GSK3004774 是一种强效的、不可吸收的 CaSR 激动剂,其 pEC50 分别为人类、小鼠和大鼠的 CaSR 为 7.3、6.6 和 6.5。GSK3004774 对人类 CaSR 的 EC50 为 50 nM。
Discription | GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR. | |||||
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Cell Research |
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目录号 | A19779 |
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分子式 | C32H40N4O3 |
分子量 | 528.69 |
CAS号 | 2138814-32-9 |
SMILES | O=C(NCCCN1CCC(C(O)=O)CC1)C(C=C2)=CC=C2N(CC3)C[C@H]3N[C@H](C)C4=CC=CC5=C4C=CC=C5 |
其他名称 | GSK 3004774, GSK-3004774 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2