GSK3395879
目录号: A19861
TRPV4 antagonist
GSK3395879 是一种选择性且可口服生物利用的瞬态受体电位香草酸受体-4(TRPV4)拮抗剂,其对 hTRPV4 的 IC50 为 1 nM。
Discription | GSK3395879 is a selective and orally bioavailable transient receptor potential vanilloid-4 (TRPV4) antagonist with an IC50 of 1 nM for hTRPV4. |
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目录号 | A19861 |
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分子式 | C20H15F4N3O5S |
分子量 | 485.41 |
CAS号 | 2215852-91-6 |
SMILES | FC1=C(C#N)C=CC(O[C@@H]2[C@@](CO)(O)CN(S(C3=C(C#N)C=C(C(F)(F)F)C=C3)(=O)=O)C2)=C1 |
其他名称 | GSK-3395879; GSK 3395879 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2