GSK5182
GSK5182 是一种高度选择性的雌激素相关受体γ（ERRγ）逆向激动剂，其 IC50 为 79 nM，并且不与其他核受体相互作用，包括 ERRα 或 ERα。
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Adooq用户使用GSK5182发表的2篇文献
生物活性
| Discription | GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα. | ||
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产品信息
| 目录号 | A19383 |
|---|---|
| 分子式 | C27H31NO3 |
| 分子量 | 417.54 |
| CAS号 | 877387-37-6 |
| SMILES | OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(O)C=C2)/C3=CC=C(OCCN(C)C)C=C3 |
| 其他名称 | GSK 5182, GSK-5182 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | 78 mg/mL | |
| Water | Insoluble | ||
| Ethanol | 78 mg/mL | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 23.95 mL | 119.75 mL | 239.5 mL |
| 0.5 mM | 4.79 mL | 23.95 mL | 47.9 mL |
| 1 mM | 2.39 mL | 11.97 mL | 23.95 mL |
| 5 mM | 0.48 mL | 2.39 mL | 4.79 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 877387-37-6 | 877387-37-6 供应商 | 877387-37-6 花费 | 877387-37-6 生产商 | 订购 877387-37-6 | 877387-37-6 代理商