GSK6853
目录号: A16330
BRPF1 bromodomain inhibitor
GSK6853 是一种强效且选择性的 BRPF1 溴结构域抑制剂。它显示出极佳的 BRPF1 效力（pKd 9.5），并且对于所有其他测试过的溴结构域具有超过1600倍的选择性。
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生物活性
| Discription | GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. shows excellent BRPF1 potency (pKd 9.5) and greater than 1600-fold selectivity over all other bromodomains tested. |
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产品信息
| 目录号 | A16330 |
|---|---|
| 分子式 | C22H27N5O3 |
| 分子量 | 409.48 |
| CAS号 | 1910124-24-1 |
| SMILES | O=C(NC1=C(N2[C@H](C)CNCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC |
| 其他名称 | GSK-6853, GSK 6853 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | Warmed: 77 mg/mL (188.04 mM) | |
| Water | Insoluble | ||
| Ethanol | Warmed: 77 mg/mL (188.04 mM) | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 24.42 mL | 122.11 mL | 244.21 mL |
| 0.5 mM | 4.88 mL | 24.42 mL | 48.84 mL |
| 1 mM | 2.44 mL | 12.21 mL | 24.42 mL |
| 5 mM | 0.49 mL | 2.44 mL | 4.88 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 1910124-24-1 | 1910124-24-1 供应商 | 1910124-24-1 花费 | 1910124-24-1 生产商 | 订购 1910124-24-1 | 1910124-24-1 代理商