H3B-5942

Name: H3B-5942
SKU: A19960
Price: 280 CNY
Rating: 5 (288 reviews)

目录号: A19960

estrogen receptor covalent 拮抗剂

H3B-5942 是一种选择性的、不可逆的、口服活性的雌激素受体共价拮抗剂，通过靶向 Cys530 来失活野生型和突变型 ERα，其 Kis 分别为 1 nM 和 0.41 nM。

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Grouped product items
规格	价格	库存
1mg	¥280.00	现货
5mg	¥735.00	现货
10mg	¥1,190.00	现货
25mg	¥2,345.00	现货
50mg	¥3,360.00	现货
100mg	¥4,480.00	现货
200mg	¥6,055.00	现货
*10mM 1mL in DMSO**	¥770.00	现货
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Data Sheet

SDS

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生物活性

Discription

H3B-5942 is a selective, irreversible and orally active estrogen receptor covalent antagonist, inactivates both wild-type and mutant ERα by targeting Cys530, with Kis of 1 nM and 0.41 nM, respectively.

Targets

Target	Value

产品信息

目录号	A19960
分子式	C31H34N4O2
分子量	494.63
CAS号	2052128-15-9
SMILES	CC/C(C1=CC=CC=C1)=C(C2=CC=C(OCCNC/C=C/C(N(C)C)=O)C=C2)\C3=CC(C=NN4)=C4C=C3
其他名称	H3B5942, H3B 5942
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro	DMSO	88 mg/mL (177.9 mM)
	Water	Insoluble
	Ethanol	12 mg/mL (24.26 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	20.22 mL	101.09 mL	202.17 mL
0.5 mM	4.04 mL	20.22 mL	40.43 mL
1 mM	2.02 mL	10.11 mL	20.22 mL
5 mM	0.4 mL	2.02 mL	4.04 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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