H3B-5942

目录号: A19960

estrogen receptor covalent antagonist

H3B-5942

H3B-5942 Chemical Structure

CAS NO. 2052128-15-9

H3B-5942 is a selective, irreversible and orally active estrogen receptor covalent antagonist, inactivates both wild-type and mutant ERα by targeting Cys530, with Kis of 1 nM and 0.41 nM, respectively.

库存: 现货

规格 价格 数量
5 mg
¥ 1,449.00
10 mg
¥ 2,499.00
50 mg
¥ 7,406.00
100 mg
¥ 14,812.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

H3B-5942 is a selective, irreversible and orally active estrogen receptor covalent antagonist, inactivates both wild-type and mutant ERα by targeting Cys530, with Kis of 1 nM and 0.41 nM, respectively.
In vitro DMSO 88 mg/mL (177.9 mM)
Water Insoluble
Ethanol 12 mg/mL (24.26 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.22 mL 101.09 mL 202.17 mL
0.5 mM 4.04 mL 20.22 mL 40.43 mL
1 mM 2.02 mL 10.11 mL 20.22 mL
5 mM 0.4 mL 2.02 mL 4.04 mL

*The above data is based on the productmolecular weight 494.63. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A19960
M. Wt 494.63
Formula C31H34N4O2
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 2052128-15-9
Synonyms H3B5942, H3B 5942
SMILES CC/C(C1=CC=CC=C1)=C(C2=CC=C(OCCNC/C=C/C(N(C)C)=O)C=C2)\C3=CC(C=NN4)=C4C=C3

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