产品详情
H3B-5942 is a selective, irreversible and orally active estrogen receptor covalent antagonist, inactivates both wild-type and mutant ERα by targeting Cys530, with Kis of 1 nM and 0.41 nM, respectively.
In vitro | DMSO | 88 mg/mL (177.9 mM) | |
Water | Insoluble | ||
Ethanol | 12 mg/mL (24.26 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 20.22 mL | 101.09 mL | 202.17 mL |
0.5 mM | 4.04 mL | 20.22 mL | 40.43 mL |
1 mM | 2.02 mL | 10.11 mL | 20.22 mL |
5 mM | 0.4 mL | 2.02 mL | 4.04 mL |
*The above data is based on the productmolecular weight 494.63. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
目录号 | A19960 |
---|---|
M. Wt | 494.63 |
Formula | C31H34N4O2 |
Purity | >99% |
Storage | Store lyophilized at -20ºC, keep desiccated. |
CAS No. | 2052128-15-9 |
Synonyms | H3B5942, H3B 5942 |
SMILES | CC/C(C1=CC=CC=C1)=C(C2=CC=C(OCCNC/C=C/C(N(C)C)=O)C=C2)\C3=CC(C=NN4)=C4C=C3 |
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