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Hesperadin是一种人极光B抑制剂，IC50为40 nM，用于防止底物磷酸化。它显著降低AMPK、Lck、MKK1、MAPKAP-K1、CHK1和PHK的活性，而不抑制MKK1在体内的活性。
靶点信息
| TbAUK1 (Cell-free assay) | Aurora B (human) (Cell-free assay) | |||
| 40 nM | 250 nM |
| In vitro (25°C) | DMSO | 100 mg/mL (193.55 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
| In vivo | 5% DMSO+40%PEG300+5% tween80+50% H2O | 2.3 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 19.35 mL | 96.77 mL | 193.54 mL |
| 0.5 mM | 3.87 mL | 19.35 mL | 38.71 mL |
| 1 mM | 1.94 mL | 9.68 mL | 19.35 mL |
| 5 mM | 0.39 mL | 1.94 mL | 3.87 mL |
*The above data is based on the productmolecular weight 516.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| 目录号 | A10448 |
|---|---|
| 作用机制 | Inhibitor (抑制剂) |
| M. Wt | 516.7 |
| Formula | C29H32N4O3S |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
| CAS No. | 422513-13-1 |
| SMILES | CCS(=O)(=O)NC1=CC\2=C(C=C1)NC(=O)/C2=C(/C3=CC=CC=C3)\NC4=CC=C(C=C4)CN5CCCCC5 |
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