I-BRD9
目录号: A15872
Selective BRD9 抑制剂
I-BRD9 是一种强效且选择性的 BRD9 抑制剂,其 pIC50 值为 7.3,而针对 BRD4 的 pIC50 值为 5.3。
Discription | I-BRD9 is a potent and selective BRD9 inhibitor with pIC50 of 7.3, while it displayed a pIC50 of 5.3 against BRD4. | ||
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Targets |
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目录号 | A15872 |
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分子式 | C22H22F3N3O3S2 |
分子量 | 497.55 |
CAS号 | 1714146-59-4 |
SMILES | N=C(C(S1)=CC2=C1C(C3=CC=CC(C(F)(F)F)=C3)=CN(CC)C2=O)NC(CC4)CCS4(=O)=O |
其他名称 | GSK602 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 94 mg/mL (188.92 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 20.1 mL | 100.49 mL | 200.98 mL |
0.5 mM | 4.02 mL | 20.1 mL | 40.2 mL |
1 mM | 2.01 mL | 10.05 mL | 20.1 mL |
5 mM | 0.4 mL | 2.01 mL | 4.02 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2