I-BRD9

Name: I-BRD9
SKU: A15872

目录号: A15872

Selective BRD9 抑制剂

I-BRD9 Chemical Structure

CAS NO. 1714146-59-4

I-BRD9是一种有效的选择性BRD9抑制剂，pIC50为7.3，而对BRD4的pIC50为5.3。

库存：现货

规格	价格	数量
5 mg	￥ 476.00
10 mg	￥ 840.00
25 mg	￥ 1,652.00

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生物活性

I-BRD9是一种有效的选择性BRD9抑制剂，pIC50为7.3，而对BRD4的pIC50为5.3。

靶点信息

BRD9	BRD4
7.3(pIC50)	5.3(pIC50)

溶解度 *

In vitro	DMSO	94 mg/mL (188.92 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	20.1 mL	100.49 mL	200.98 mL
0.5 mM	4.02 mL	20.1 mL	40.2 mL
1 mM	2.01 mL	10.05 mL	20.1 mL
5 mM	0.4 mL	2.01 mL	4.02 mL

*The above data is based on the productmolecular weight 497.55. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15872
作用机制	Inhibitor (抑制剂)
M. Wt	497.55
Formula	C22H22F3N3O3S2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1714146-59-4
Synonyms	GSK602
SMILES	N=C(C(S1)=CC2=C1C(C3=CC=CC(C(F)(F)F)=C3)=CN(CC)C2=O)NC(CC4)CCS4(=O)=O