I-CBP112

Name: I-CBP112
SKU: A13165

目录号: A13165

CBP/p300 bromodomain 抑制剂

I-CBP112 Chemical Structure

CAS NO. 1640282-31-0

I-CBP112是一种高效且选择性的p300/CBP溴结构域抑制剂（对于CBP，IC50为?0.14-0.17 uM，对于p300为?0.625 uM）。

库存：现货

规格	价格	数量
10 mg	￥ 1,050.00
25 mg	￥ 2,100.00
50 mg	￥ 3,500.00

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生物活性

I-CBP112是一种高效且选择性的p300/CBP溴结构域抑制剂（对于CBP，IC50为?0.14-0.17 uM，对于p300为?0.625 uM）。

溶解度 *

In vitro	DMSO	86 mg/mL (183.53 mM)
	Water	86 mg/mL (183.53 mM)
	Ethanol	86 mg/mL (183.53 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.34 mL	106.7 mL	213.41 mL
0.5 mM	4.27 mL	21.34 mL	42.68 mL
1 mM	2.13 mL	10.67 mL	21.34 mL
5 mM	0.43 mL	2.13 mL	4.27 mL

*The above data is based on the productmolecular weight 468.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A13165
作用机制	Inhibitor (抑制剂)
M. Wt	468.59
Formula	C27H36N2O5
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1640282-31-0
Synonyms	ICBP112
SMILES	CCC(=O)N1CCOC2=C(C1)C=C(C=C2OC[C@H]3CCCN(C3)C)C4=CC(=C(C=C4)OC)OC