I-CBP112
目录号: A13165
CBP/p300 bromodomain 抑制剂
I-CBP112 是一种高效且选择性的 p300/CBP 溴结构域抑制剂(CBP 的 IC50 约为 0.14-0.17 uM,p300 的 IC50 约为 0.625 uM)。
Discription | I-CBP112 is a highly potent and selective p300/CBP bromodomain inhibitor (IC50 ~0.14-0.17 uM for CBP and ~0.625 uM for p300). | |||||
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Cell Research |
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目录号 | A13165 |
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分子式 | C27H36N2O5 |
分子量 | 468.59 |
CAS号 | 1640282-31-0 |
SMILES | CCC(=O)N1CCOC2=C(C1)C=C(C=C2OC[C@H]3CCCN(C3)C)C4=CC(=C(C=C4)OC)OC |
其他名称 | ICBP112 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 86 mg/mL (183.53 mM) | |
Water | 86 mg/mL (183.53 mM) | ||
Ethanol | 86 mg/mL (183.53 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 21.34 mL | 106.7 mL | 213.41 mL |
0.5 mM | 4.27 mL | 21.34 mL | 42.68 mL |
1 mM | 2.13 mL | 10.67 mL | 21.34 mL |
5 mM | 0.43 mL | 2.13 mL | 4.27 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2