IDO/TDO-IN-1
目录号: A18566
IDO/TDO dual 抑制剂
IDO/TDO-IN-1 是一种高效的口服活性双重吲哚胺-2,3-双加氧酶(IDO)和色氨酸-2,3-双加氧酶(TDO)抑制剂,其半抑制浓度(IC50)分别为9.7纳摩尔和47纳摩尔。
Discription | IDO/TDO-IN-1 is a highly potent and orally active dual indoleamine-2,3-dioxygenase (IDO) and tryptophan 2,3-dioxygenase (TDO) inhibitor with IC50s of 9.7 and 47 nM, respectively . | |||||
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Cell Research |
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目录号 | A18566 |
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分子式 | C25H24FN5 |
分子量 | 413.49 |
CAS号 | 2033173-01-0 |
SMILES | CN1N=CC(C2=CC=C(N3CCC([C@@H](C4=C5C=CC=C4F)N6C5=CN=C6)CC3)C=C2)=C1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2