Imidafenacin
目录号: A15490
M3 receptors 抑制剂
Imidafenacin 是一种强效且选择性的 M3 受体 抑制剂,其Kb值为0.317 nM;对 M2 受体 的抑制作用较弱(IC50=4.13 nM)。
Discription | Imidafenacin is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors(IC50=4.13 nM). |
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目录号 | A15490 |
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分子式 | C20H21N3O |
分子量 | 319.4 |
CAS号 | 170105-16-5 |
SMILES | CC1=NC=CN1CCC(C2=CC=CC=C2)(C3=CC=CC=C3)C(=O)N |
其他名称 | KRP-197, ONO-8025 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 60 mg/mL (187.85 mM) | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 31.31 mL | 156.54 mL | 313.09 mL |
0.5 mM | 6.26 mL | 31.31 mL | 62.62 mL |
1 mM | 3.13 mL | 15.65 mL | 31.31 mL |
5 mM | 0.63 mL | 3.13 mL | 6.26 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2