Imidafenacin

Name: Imidafenacin
SKU: A15490

目录号: A15490

M3 receptors 抑制剂

Imidafenacin Chemical Structure

CAS NO. 170105-16-5

Imidafenacin是一种有效的选择性M3受体抑制剂，Kb为0.317 nM。对M2受体的效力较低（IC50 = 4.13 nM）。

库存：现货

规格	价格	数量
10 mg	￥ 315.00
25 mg	￥ 630.00
50 mg	￥ 1,085.00
100 mg	￥ 1,855.00

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生物活性

Imidafenacin是一种有效的选择性M3受体抑制剂，Kb为0.317 nM。对M2受体的效力较低（IC50 = 4.13 nM）。

溶解度 *

In vitro	DMSO	60 mg/mL (187.85 mM)
	* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	31.31 mL	156.54 mL	313.09 mL
0.5 mM	6.26 mL	31.31 mL	62.62 mL
1 mM	3.13 mL	15.65 mL	31.31 mL
5 mM	0.63 mL	3.13 mL	6.26 mL

*The above data is based on the productmolecular weight 319.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15490
作用机制	Inhibitor (抑制剂)
M. Wt	319.4
Formula	C20H21N3O
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	170105-16-5
Synonyms	KRP-197, ONO-8025
SMILES	CC1=NC=CN1CCC(C2=CC=CC=C2)(C3=CC=CC=C3)C(=O)N