Immethridine hydrobromide
目录号: A13641
histamine H3 receptor 激动剂
Immethridine hydrobromide 是一种强效且高度选择性的组胺 H3 受体激动剂(pEC50 = 9.74),相较于 H4 受体 具有 300 倍的选择性(pKi 值分别为 9.07 和 6.61)。
Discription | Immethridine hydrobromide is a strong and highly selective histamine H3 receptor agonist (pEC50 = 9.74) that displays 300-fold selectivity over the H4 receptor (pKi values are 9.07 and 6.61 respectively). |
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目录号 | A13641 |
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分子式 | C9H9N3.HBr |
分子量 | 240.103 |
CAS号 | 87976-03-2 |
SMILES | C1=CN=CC=C1CC2=CN=CN2.Br |
其他名称 | Immethridine HBr |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2