JQEZ5
目录号: A16961
EZH2 抑制剂
JQEZ5 是一种强效且选择性的 SAM-竞争性 EZH2 赖氨酸甲基转移酶抑制剂,其 IC50 值为 11 nM。
Discription | JQEZ5 is a potent and selective SAM-competitive EZH2 lysine methyltransferase inhibitor with IC50 value of 11 nM. | ||
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目录号 | A16961 |
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分子式 | C30H38N8O2 |
分子量 | 542.68 |
CAS号 | 1913252-04-6 |
SMILES | CC(C)N1N=CC2=C(C=C(N=C12)C3=CC=C(N4CCN(CC4)C)N=C3)C(NCC5=C(CCC)C=C(C)NC5=O)=O |
其他名称 | JQEZ-5, JQEZ 5, JQ-EZ-05, JQ-EZ05, JQ-EZ 05 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2