Ketanserin (Vulketan Gel)
目录号: A10497
5-HT2A serotonin receptor 拮抗剂
Ketanserin(Vulketan Gel)是一种特异性 5-HT2A 血清素受体拮抗剂,其对大鼠和人类 5-HT2A 的Ki值为2.5 nM。
Discription | Ketanserin (Vulketan Gel) is specific 5-HT2A serotonin receptor antagonist with a Ki of 2.5 nM for rat and human 5-HT2A. | |||||
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Cell Research |
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目录号 | A10497 |
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分子式 | C22H22FN3O3 |
分子量 | 395.43 |
CAS号 | 74050-98-9 |
SMILES | C1CN(CCC1C(=O)C2=CC=C(C=C2)F)CCN3C(=O)C4=CC=CC=C4NC3=O |
其他名称 | R 41468, Vulketan Gel |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 2 mg/mL (5.05 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
In vivo | 4% DMSO+40% PEG 300+4% Tween 80+ddH2O | 1 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 25.29 mL | 126.44 mL | 252.89 mL |
0.5 mM | 5.06 mL | 25.29 mL | 50.58 mL |
1 mM | 2.53 mL | 12.64 mL | 25.29 mL |
5 mM | 0.51 mL | 2.53 mL | 5.06 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2