Ketanserin (Vulketan Gel)

Name: Ketanserin (Vulketan Gel)
SKU: A10497

目录号: A10497

5-HT2A serotonin receptor 拮抗剂

Ketanserin (Vulketan Gel) Chemical Structure

CAS NO. 74050-98-9

Ketanserin (Vulketan Gel)是大鼠和人5-HT2A血清素受体拮抗剂，Ki为2.5 nM。

库存：现货

规格	价格	数量
50 mg	￥ 280.00
100 mg	￥ 420.00
250 mg	￥ 840.00
500 mg	￥ 1,540.00

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产品仅用于科学研究，不针对患者销售，望谅解.

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生物活性

Ketanserin (Vulketan Gel)是大鼠和人5-HT2A血清素受体拮抗剂，Ki为2.5 nM。

靶点信息

5-HT2A	5-HT2C (Rat)	5-HT2C (Human)
2.5 nM(Ki)	50 nM(Ki)	100 nM(Ki)

溶解度 *

In vitro (25°C)	DMSO	2 mg/mL (5.05 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	4% DMSO+40% PEG 300+4% Tween 80+ddH2O	1 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	25.29 mL	126.44 mL	252.89 mL
0.5 mM	5.06 mL	25.29 mL	50.58 mL
1 mM	2.53 mL	12.64 mL	25.29 mL
5 mM	0.51 mL	2.53 mL	5.06 mL

*The above data is based on the productmolecular weight 395.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A10497
作用机制	Antagonist (拮抗剂)
M. Wt	395.43
Formula	C22H22FN3O3
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	74050-98-9
Synonyms	R 41468, Vulketan Gel
SMILES	C1CN(CCC1C(=O)C2=CC=C(C=C2)F)CCN3C(=O)C4=CC=CC=C4NC3=O