KPT 9274 (ATG-019)

Name: KPT 9274 (ATG-019)
SKU: A15506
Price: 350 CNY
Rating: 5 (288 reviews)

目录号: A15506

PAK4/NAMPT 抑制剂

KPT 9274（ATG-019）是一种口服生物利用度高的小分子药物，它是PAK4和NAMPT的非竞争性双重抑制剂。在无细胞酶活性测定中，其对NAMPT的IC50约为120纳摩尔。

Skip to the end of the images gallery

Skip to the beginning of the images gallery

Grouped product items
规格	价格	库存
1mg	¥350.00	现货
2mg	¥665.00	现货
5mg	¥980.00	现货
10mg	¥1,610.00	现货
25mg	¥2,730.00	现货
50mg	¥3,920.00	现货
100mg	¥5,390.00	现货
*10mM 1mL in DMSO**	¥1,330.00	现货
更大包装	更多折扣

大包装询价

Notify me when the price drops

全国免运费, 顺丰次日达

重要通知：仅供研究使用。我们不向患者销售。

Data Sheet

SDS

顾客使用 Adooq 产品发表的高质量科研文献

生物活性

Discription	KPT 9274 ( ATG-019) is an orally bioavailable small molecule that is a non-competitive dual inhibitor of PAK4 and NAMPT. It shows an IC50 of ~120 nM for NAMPT in a cell-free enzymatic assay.

产品信息

目录号	A15506
分子式	C35H29F3N4O3
分子量	610.63
CAS号	1643913-93-2
SMILES	FC1=CC=C(C2=CC(C3=CC=C(C(N4CCC(F)(F)CC4)=O)C=C3)=CC5=C2OC(C/N=C(O)/C([H])=C([H])/C6=NC(N)=CC=C6)=C5)C=C1
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro	DMSO	85 mg/mL (139.2 mM)
	Water	Insoluble
	Ethanol	85 mg/mL (139.2 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	16.38 mL	81.88 mL	163.77 mL
0.5 mM	3.28 mL	16.38 mL	32.75 mL
1 mM	1.64 mL	8.19 mL	16.38 mL
5 mM	0.33 mL	1.64 mL	3.28 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

Calculate Reset

* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Keywords: 购买 KPT 9274 (ATG-019) | KPT 9274 (ATG-019) 供应商 | KPT 9274 (ATG-019) 花费 | KPT 9274 (ATG-019) 生产商 | 订购 KPT 9274 (ATG-019) | KPT 9274 (ATG-019) 代理商 | 购买 1643913-93-2 | 1643913-93-2 供应商 | 1643913-93-2 花费 | 1643913-93-2 生产商 | 订购 1643913-93-2 | 1643913-93-2 代理商