L-371,257
目录号: A21219
oxytocin receptor 拮抗剂
L-371,257 是一种口服生物利用度高的、不穿透血脑屏障的、选择性和竞争性的催产素受体拮抗剂(pA2=8.4),在催产素受体(Ki=19 nM)和抗利尿激素V1a受体(Ki=3.7 nM)上具有高亲和力。
Discription | L-371,257 is an orally bioavailable, non-blood-brain barrier penetrant, selective and competitive antagonist of oxytocin receptor (pA2=8.4) with high affinity at both the oxytocin receptor (Ki=19 nM) and vasopressin V1a receptor (Ki=3.7 nM). | |||||
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Cell Research |
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目录号 | A21219 |
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分子式 | C28H33N3O6 |
分子量 | 507.58 |
CAS号 | 162042-44-6 |
SMILES | O=C(OC1)N(C2CCN(C(C3=C(OC)C=C(OC4CCN(C(C)=O)CC4)C=C3)=O)CC2)C5=C1C=CC=C5 |
其他名称 | L-371257, L371,257, L371257 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2