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Iptacopan (LNP023)

目录号: A18905
Factor B 抑制剂
LNP023 是一种高效的因子 B(FB)抑制剂,其 IC50 值为 10 nM。LNP023 显示出对人类 FB 的直接、可逆和高亲和力结合(KD=7.9 nM)。
Grouped product items
规格 价格 库存 数量
1mg
¥875.00
现货
5mg
¥1,050.00
现货
10mg
¥1,785.00
现货
25mg
¥3,255.00
现货
50mg
¥5,460.00
现货
100mg
¥9,135.00
现货
500mg
¥33,705.00
现货
10mM * 1mL in DMSO
¥2,485.00
现货
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重要通知:仅供研究使用。我们不向患者销售。

顾客使用 Adooq 产品发表的高质量科研文献
Adooq用户使用Iptacopan (LNP023)发表的1篇文献
  • Wenbin Yang, .et al. , J Clin Invest, 2022, Oct 17;132(20):e157975 PMID: 36250462
  • 生物活性
    Discription LNP023 is a highly potent factor B (FB) inhibitor with an IC50 value of 10 nM. LNP023 shows direct, reversible, and high-affinity binding to human FB (KD=7.9 nM).
    产品信息
    目录号 A18905
    分子式 C25H30N2O4
    分子量 422.52
    CAS号 1644670-37-0
    SMILES O=C(O)C1=CC=C([C@H]2N(CC3=C(OC)C=C(C)C4=C3C=CN4)CC[C@H](OCC)C2)C=C1
    其他名称 LNP 023, LNP-023
    储存条件

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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