Lurasidone (SM13496)
目录号: A11214
Dopamine D2 抑制剂
Lurasidone 是一种非典型抗精神病药物,它可以缓解阳性症状(例如,幻觉、妄想),尽管其具有强大的 D2受体拮抗作用,但除了静坐不能症外,不会引起锥体外系副作用。
Discription | Lurasidone is an atypical antipsychotic that alleviates positive symptoms (e.g., hallucinations, delusions) without inducing extrapyramidal side effects except for akathisia,despite its potent D2 antagonistic actions. | ||
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目录号 | A11214 |
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分子式 | C28H36N4O2S |
分子量 | 492.7 |
CAS号 | 367514-87-2 |
SMILES | C1CC[C@H]([C@@H](C1)CN2CCN(CC2)C3=NSC4=CC=CC=C43)CN5C(=O)[C@H]6[C@@H]7CC[C@@H](C7)[C@H]6C5=O |
其他名称 | SM13496, SM-13496, SM 13496 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 7 mg/mL (14.2 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 20.3 mL | 101.48 mL | 202.96 mL |
0.5 mM | 4.06 mL | 20.3 mL | 40.59 mL |
1 mM | 2.03 mL | 10.15 mL | 20.3 mL |
5 mM | 0.41 mL | 2.03 mL | 4.06 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2