LY 2183240
目录号: A11960
FAAH inhibitor
LY 2183240 既是内源性大麻素苯丙酰胺的强效抑制剂,也是脂肪酰胺水解酶(FAAH)的抑制剂,后者是负责降解苯丙酰胺的主要酶。
Discription | LY 2183240 acts both as a potent inhibitor of the reuptake of the endocannabinoid anandamide, and as an inhibitor of fatty acid amide hydrolase (FAAH), the primary enzyme responsible for degrading anandamide. | |||||
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Cell Research |
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目录号 | A11960 |
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分子式 | C17H17N5O |
分子量 | 307.35 |
CAS号 | 874902-19-9 |
SMILES | CN(C)C(=O)N1C(=NN=N1)CC2=CC=C(C=C2)C3=CC=CC=C3 |
其他名称 | LY2183240, LY-2183240 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 56 mg/mL (182.2 mM) | |
Water | Insoluble | ||
Ethanol | 56 mg/mL | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 32.54 mL | 162.68 mL | 325.36 mL |
0.5 mM | 6.51 mL | 32.54 mL | 65.07 mL |
1 mM | 3.25 mL | 16.27 mL | 32.54 mL |
5 mM | 0.65 mL | 3.25 mL | 6.51 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2