LY-2940094
目录号: A19125
NOP receptor antagonist
LY-2940094 是一种强效、选择性且可口服的伤害素受体(NOP受体)拮抗剂,具有高亲和力(Ki=0.105 nM)和拮抗效力(Kb=0.166 nM)。LY-2940094 在动物模型中降低乙醇自我给药。
Discription | LY-2940094 is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY-2940094 reduces ethanol self-administration in animal models. |
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目录号 | A19125 |
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分子式 | C22H23ClF2N4O2S |
分子量 | 480.96 |
CAS号 | 1307245-86-8 |
SMILES | OCC1=CC=CN=C1N2N=C(C)C(CN3CCC4(C5=C(C=C(Cl)S5)C(F)(F)CO4)CC3)=C2 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2