Mcl-1-PUMA Modulator-8
目录号: A18369
Mcl-1-PUMA interface 抑制剂
Mcl1-IN-8(Comp8)是一种 Mcl-1-PUMA 界面抑制剂,其Ki值为0.3 μM。Mcl1-IN-8(Comp8)在减少 PUMA 依赖性凋亡的同时,能够抑制癌细胞中 Mcl-1 介导的抗凋亡活性。
Discription | Mcl1-IN-8 (Comp8) is a Mcl-1-PUMA interface inhibitor, with a Ki of 0.3 μM. Mcl1-IN-8 (Comp8) exhibits dual activity on reduce PUMA-dependent apoptosis while deactivating Mcl-1-mediated anti-apoptosis in cancer cells. | ||
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目录号 | A18369 |
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分子式 | C22H23N3O2S |
分子量 | 393.51 |
CAS号 | 678158-55-9 |
SMILES | O=C1N=C(N2CCN(CCO)CC2)S/C1=C\C3=CC=C(C4=CC=CC=C4)C=C3 |
其他名称 | Mcl-1-PUMA modulator-8 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2