MK-3207
目录号: A15165
CGRP Receptor 拮抗剂
MK-3207 是一种强效且可口服的 CGRP 受体拮抗剂(IC50= 0.12 nM;Ki 值= 0.024 nM);与人类 AM1、AM2、CTR 和 AMY3 相比具有高度选择性。
Discription | MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki value= 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3. | |||||
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Cell Research |
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目录号 | A15165 |
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分子式 | C31H29F2N5O3 |
分子量 | 557.59 |
CAS号 | 957118-49-9 |
SMILES | C1CCC2(C1)C(=O)N(C(CN2)C3=CC(=CC(=C3)F)F)CC(=O)NC4=CC5=C(CC6(C5)C7=C(NC6=O)N=CC=C7)C=C4 |
其他名称 | MK3207, MK 3207 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2