MK-571 sodium salt

Name: MK-571 sodium salt
SKU: A15983

目录号: A15983

CysLT1 receptor 拮抗剂

MK-571 sodium salt Chemical Structure

CAS NO. 115103-85-0

MK-571 sodium salt是一种选择性的口服活性CysLT1受体拮抗剂。它阻断LTD4而不是LTC4与人和豚鼠肺膜的结合，Ki值分别为0.22 nM和2.1 nM。

库存：现货

规格	价格	数量
5 mg	￥ 315.00
10 mg	￥ 560.00
50 mg	￥ 2,240.00

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生物活性

MK-571 sodium salt是一种选择性的口服活性CysLT1受体拮抗剂。它阻断LTD4而不是LTC4与人和豚鼠肺膜的结合，Ki值分别为0.22 nM和2.1 nM。

靶点信息

CysLT1	MRP1	MRP4	cMOAT

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	18.62 mL	93.1 mL	186.2 mL
0.5 mM	3.72 mL	18.62 mL	37.24 mL
1 mM	1.86 mL	9.31 mL	18.62 mL
5 mM	0.37 mL	1.86 mL	3.72 mL

*The above data is based on the productmolecular weight 537.06. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15983
作用机制	Antagonist (拮抗剂)
M. Wt	537.06
Formula	C26H26ClN2NaO3S2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	115103-85-0
Synonyms	L-660,711, L660,711, L 660,711, L-660711
SMILES	O=C([O-])CCSC(C1=CC=CC(/C=C/C2=NC3=CC(Cl)=CC=C3C=C2)=C1)SCCC(N(C)C)=O.[Na+]