MK-6096 (Filorexant)

Name: MK-6096 (Filorexant)
SKU: A13168
Price: 175 CNY
Rating: 5 (288 reviews)

目录号: A13168

Orexin receptor 拮抗剂

MK6096，也被称为filorexant，是一种口服生物利用度高的强效且选择性的可逆OX(1)R和OX(2)R拮抗剂，目前正处于失眠症的临床开发阶段。MK-6096展示了对人类OX(1)R和OX(2)R的强效结合和拮抗作用（结合力<3 nM，FLIPR中11 nM），并且在超过170种受体和酶的检测中没有显著的非目标活性。

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Grouped product items
规格	价格	库存
1mg	¥175.00	现货
5mg	¥420.00	现货
10mg	¥770.00	现货
25mg	¥1,330.00	现货
50mg	¥2,030.00	现货
100mg	¥3,010.00	现货
*10mM 1mL in DMSO**	¥490.00	现货
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Data Sheet

SDS

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生物活性

Discription

MK6096, also known as filorexant, is an orally bioavailable potent and selective reversible antagonist of OX(1)R and OX(2)R currently in clinical development for insomnia. MK-6096 demonstrated potent binding and antagonism of both human OX(1)R and OX(2)R (<3 nM in binding, 11 nM in FLIPR), with no significant off-target activities against a panel of >170 receptors and enzymes.

Cell Research

Cell Line	Type	Value	Description	References

产品信息

目录号	A13168
分子式	C24H25FN4O2
分子量	420.48
CAS号	1088991-73-4
SMILES	CC1=CC=C(C2=NC=CC=N2)C(C(N3C[C@@H](COC4=NC=C(F)C=C4)CC[C@@H]3C)=O)=C1
其他名称	MK6096, MK-6096, MK 6096
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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