ML-3043
目录号: A12408
p38 MAPK 抑制剂
ML-3043 是一种 p38 MAPK 抑制剂(IC50 = 0.38 μM)。在外周血单核细胞(PBMC)实验中抑制 IL-1β 和 TNF-α 的释放(IC50 值分别为 0.039 和 0.16 μM)。
Discription | ML-3043 is a p38 MAPK inhibitor (IC50 = 0.38 μM). Inhibits the release of IL-1β and TNF-α in a peripheral blood mononuclear cell (PBMC) assay (IC50 values are 0.039 and 0.16 μM respectively). |
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目录号 | A12408 |
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分子式 | C23H21FN4S |
分子量 | 404.5 |
CAS号 | 549505-65-9 |
SMILES | CC(C1=CC=CC=C1)NC2=NC=CC(=C2)C3=C(NC(=N3)SC)C4=CC=C(C=C4)F |
其他名称 | ML3043, ML 3043 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2