Mozavaptan
目录号: A16622
nonpeptide vasopressin V2 receptor 拮抗剂
Mozavaptan(OPC31260)是一种口服有效的非肽类抗利尿激素V2受体拮抗剂,其IC50为14 nM。
Discription | Mozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM. | |||||
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Cell Research |
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目录号 | A16622 |
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分子式 | C27H29N3O2 |
分子量 | 427.54 |
CAS号 | 137975-06-5 |
SMILES | CC1=CC=CC=C1C(NC2=CC=C(C(N3C(C=CC=C4)=C4C(N(C)C)CCC3)=O)C=C2)=O |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 1 mg/mL (2.33 mM) | |
Water | Insoluble | ||
Ethanol | 1 mg/mL (2.33 mM) | ||
In vivo | 30% propylene glycol, 5% Tween 80, 65% D5W | 28 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 23.39 mL | 116.95 mL | 233.9 mL |
0.5 mM | 4.68 mL | 23.39 mL | 46.78 mL |
1 mM | 2.34 mL | 11.69 mL | 23.39 mL |
5 mM | 0.47 mL | 2.34 mL | 4.68 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2