MPEP
目录号: A12589
mGlu5 receptor 拮抗剂
MPEP 是一种强效且高度选择性的非竞争性拮抗剂，针对 mGlu5 受体亚型（IC50 = 36 nM），同时也是 mGlu4 受体的正向异构调节剂。
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生物活性
| Discription | MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors. | |||||
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| Targets |
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| Cell Research |
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产品信息
| 目录号 | A12589 |
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| 分子式 | C14H11N |
| 分子量 | 193.249 |
| CAS号 | 96206-92-7 |
| SMILES | CC1=CC=CC(=N1)C#CC2=CC=CC=C2 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro (25°C) | DMSO | 36 mg/mL (186.3 mM) | |
| Water | Insoluble | ||
| Ethanol | 36 mg/mL (186.3 mM) | ||
| In vivo | 2% DMSO+30% PEG 300+5% Tween 80 | 9 mg/mL | |
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 51.75 mL | 258.73 mL | 517.47 mL |
| 0.5 mM | 10.35 mL | 51.75 mL | 103.49 mL |
| 1 mM | 5.17 mL | 25.87 mL | 51.75 mL |
| 5 mM | 1.03 mL | 5.17 mL | 10.35 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 96206-92-7 | 96206-92-7 供应商 | 96206-92-7 花费 | 96206-92-7 生产商 | 订购 96206-92-7 | 96206-92-7 代理商