MRS1706
目录号: A16868
adenosine A2B receptor 激动剂
MRS1706 是一种选择性的腺苷 A2B 受体反向激动剂,其对人类 A2B、A1、A2A 和 A3 受体的 Ki 值分别为 1.39、157、112 和 230 nM。
Discription | MRS1706 is a selective adenosine A2B receptor inverse agonist with Ki values of 1.39, 157, 112, and 230 nM for human A2B, A1, A2A, and A3 receptors, respectively. |
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目录号 | A16868 |
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分子式 | C27H29N5O5 |
分子量 | 503.56 |
CAS号 | 264622-53-9 |
SMILES | O=C(NC1=CC=C(C(C)=O)C=C1)COC2=CC=C(C(N3)=NC(N(CCC)C(N4CCC)=O)=C3C4=O)C=C2 |
其他名称 | MRS 1706, MRS-1706 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2