Naproxen etemesil
目录号: A13052
COX-1 and COX-2 抑制剂
纳普洛昔林依替米松是一种亲脂性、非酸性的无活性前体药物,它在被吸收后通过水解转化为药理活性的纳普洛昔林。纳普洛昔林是一种COX-1 和 COX-2 抑制剂,在细胞实验中的IC50分别为8.72和5.15微摩尔。
Discription | Naproxen etemesil is a lipophilic, non-acidic, inactive prodrug of naproxen that is hydrolysed to pharmacologically active Naproxen once absorbed. Naproxen is a COX-1 and COX-2 inhibitor with IC50s of 8.72 and 5.15 μM, respectively in cell assay. |
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目录号 | A13052 |
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分子式 | C17H20O5S |
分子量 | 336.4 |
CAS号 | 385800-16-8 |
SMILES | O=C(OCCS(C)(=O)=O)[C@@H](C)C1=CC2=CC=C(OC)C=C2C=C1 |
其他名称 | LT-NS 001; MX 1094, MX-1094, MX1094 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2