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￥ 0.00 Neuronal Signaling
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(+)-Bicuculline
Catalog No. A12590 -
AWD 131-138
Catalog No. A13726 -
2-Hydroxysaclofen
Catalog No. A13696 -
Cloflubicyne
Catalog No. A13932 -
a5IA
Catalog No. A14343 -
Guvacine hydrochloride
Catalog No. A13613 GABA uptake 抑制剂Guvacine hydrochloride可抑制GABA的摄取（hGABA T-1，rGABA T-2，hGABA T-3和hBGT-1的IC50值分别为14、58、119和1870 uM）。 了解更多 -
Muscimol hydrobromide
Catalog No. A13459 GABA(A) receptor 激动剂Muscimol hydrobromide是抗抑郁药氟西汀的活性代谢产物，可抑制5-羟色胺的摄取，pKi值为7.35.1。诺氟西汀的S-对映体的5-羟色胺再摄取阻断效能比R-对映体高20倍（分别为pKis = 7.86与6.51）。 了解更多 -
Etifoxine
Catalog No. A15083 -
Etifoxine hydrochloride
Catalog No. A15084 -
Picrotoxin
Catalog No. A14004 GABAA receptor 拮抗剂Picrotoxin是GABAA受体拮抗剂。该化合物已显示可增加下丘脑的去甲肾上腺素水平和周转率。 了解更多 -
Tiagabine hydrochloride
Catalog No. A16135 -
Piperazine
Catalog No. A16171 -
Lorediplon
Catalog No. A13449 -
(-)-Securinine
Catalog No. A17102 GABA receptor 拮抗剂(-)-Securinine是一种最初从S. suffructicosa分离的生物碱。Securinine是一种特定的GABA受体拮抗剂，已发现在体内具有显着的CNS活性。 了解更多 -
Afloqualone
Catalog No. A17276 GABA receptor agonistAfloqualone, also known as HQ-495, is a centrally acting muscle relaxant. Afloqualone inhibits vestibular nystagmus probably due to both inhibition of selective polysynaptic transmission and enhancement of the effects of GABA and glycine in the lateral vestibular nucleus (LVN), and its GABA-enhancing effect is thought to be attributable to the increased sensitivity of GABA receptors of the LVN neuron site. 了解更多 -
Homotaurine
Catalog No. A17944 GABA receptor agonistTramiprosate, also known as homotaurine, is a gamma-Aminobutyric acid (GABA) receptor agonist and a glycosaminoglycan mimetic used in the treatment of Alzheimer's disease. 了解更多 -
Baclofen
Catalog No. A18248 GABA agonistBaclofen is a GABA agonist specific for GABA-B receptors. Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing It acts at spinal and supraspinal sites, reducing excitatory transmission. 了解更多 -
Flupirtine maleate
Catalog No. A10251 NMDA 拮抗剂Flupirtine maleate是Flupirine的盐形式，是一种非阿片类中枢性镇痛药，是一种选择性的神经元钾离子通道开放剂，也具有NMDA受体拮抗剂特性。 了解更多 -
TCN 201
Catalog No. A11947 -
SDZ 220-581
Catalog No. A12426 -
(-)-MK 801 maleate
Catalog No. A13435 NMDA receptor 拮抗剂.(-)-MK 801 maleate是一种有效的、选择性的、非竞争性的NMDA受体拮抗剂。它通过与NMDA相关离子通道内的一个位点结合而起作用。 了解更多 -
SDZ 220-581 Ammonium salt
Catalog No. A15235 -
L-701324
Catalog No. A15522 -
(+)-MK 801 Maleate
Catalog No. A12761 -
GV-196771A
Catalog No. A13438 NMDA receptor antagonistGV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. 了解更多 -
Ifenprodil tartrate
Catalog No. A16583 NMDA receptor antagonistIfenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). 了解更多 -
Transcrocetinate disodium
Catalog No. A21051 NMDA receptor antagonistTranscrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. 了解更多 -
MDL 105519
Catalog No. A21192 NMDA receptor antagonistMDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. 了解更多
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