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￥ 0.00 Neuronal Signaling
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Flumazenil
Catalog No. A10397 Benzodiazepine 拮抗剂Flumazenil是竞争性抑制GABA/苯二氮卓受体复合物上苯二氮卓识别位点的活性。Flumazenil在一些活性动物模型中是弱部分激动剂，但在人类中很少或没有激动剂活性。 了解更多 -
(+)-Bicuculline
Catalog No. A12590 -
2-Hydroxysaclofen
Catalog No. A13696 -
Cloflubicyne
Catalog No. A13932 -
Picrotoxin
Catalog No. A14004 GABAA receptor 拮抗剂Picrotoxin是GABAA受体拮抗剂。该化合物已显示可增加下丘脑的去甲肾上腺素水平和周转率。 了解更多 -
(-)-Securinine
Catalog No. A17102 GABA receptor 拮抗剂(-)-Securinine是一种最初从S. suffructicosa分离的生物碱。Securinine是一种特定的GABA受体拮抗剂，已发现在体内具有显着的CNS活性。 了解更多 -
Flupirtine maleate
Catalog No. A10251 NMDA 拮抗剂Flupirtine maleate是Flupirine的盐形式，是一种非阿片类中枢性镇痛药，是一种选择性的神经元钾离子通道开放剂，也具有NMDA受体拮抗剂特性。 了解更多 -
TCN 201
Catalog No. A11947 -
SDZ 220-581
Catalog No. A12426 -
(-)-MK 801 maleate
Catalog No. A13435 NMDA receptor 拮抗剂.(-)-MK 801 maleate是一种有效的、选择性的、非竞争性的NMDA受体拮抗剂。它通过与NMDA相关离子通道内的一个位点结合而起作用。 了解更多 -
SDZ 220-581 Ammonium salt
Catalog No. A15235 -
L-701324
Catalog No. A15522 -
(+)-MK 801 Maleate
Catalog No. A12761 -
GV-196771A
Catalog No. A13438 NMDA receptor antagonistGV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. 了解更多 -
Ifenprodil tartrate
Catalog No. A16583 NMDA receptor antagonistIfenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). 了解更多 -
Transcrocetinate disodium
Catalog No. A21051 NMDA receptor antagonistTranscrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. 了解更多 -
MDL 105519
Catalog No. A21192 NMDA receptor antagonistMDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. 了解更多 -
Radiprodil
Catalog No. A21193 NMDA NR2B antagonistRadiprodil (RGH-896) is an orally active and selective NMDA NR2B antagonist. A potential therapeutic agent in treatment of neuropathic pain and possibly other chronic pain conditions. 了解更多 -
7-Chlorokynurenic acid sodium salt
Catalog No. A21879 NMDA receptor antagonist7-Chlorokynurenic acid sodium salt is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM). 了解更多 -
SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581
Catalog No. A21897 NMDA receptor antagonistSDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. 了解更多 -
Rislenemdaz
Catalog No. A21907 NMDA receptor GluN2B antagonistRislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. 了解更多 -
Memantine hydrochloride
Catalog No. A11708 NMDA receptor 拮抗剂Memantine hydrochloride是nmda受体的拮抗剂，与离子通道位点结合。它还是CYP2B6和CYP2D6抑制剂，作用于重组CYP2B6和CYP2D6，Ki分别为0.51 nM和94.9 μM。它被用于治疗帕金森综合征。 了解更多 -
Orphenadrine citrate
Catalog No. A11712 -
NVP-AAM077 Tetrasodium Hydrate (PEAQX)
Catalog No. A14071 -
D-AP5
Catalog No. A17044 -
Mephenesin
Catalog No. A17493 NMDA receptor antagonistMephenesin is an NMDA receptor antagonist, is a centrally acting muscle relaxant. 了解更多 -
Phenoxybenzamine hydrochloride
Catalog No. A10719 α-adrenergic (AR) 拮抗剂/CaM 抑制剂Phenoxybenzamine hydrochloride是一种细胞可渗透的，非特异性的，不可逆的α-肾上腺素（AR）拮抗剂，也可作为CaM抑制剂。 了解更多 -
Fesoterodine fumarate (Toviaz)
Catalog No. A10386 -
5-hydroxymethyl tolterodine (PNU 200577)
Catalog No. A11166 muscarinic receptor 拮抗剂5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物，tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。 了解更多 -
Rocuronium bromide
Catalog No. A10803 -
Biperiden HCl
Catalog No. A10147 -
Tolterodine tartrate (Detrol LA)
Catalog No. A10937
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- Purinergic (P2Y) Receptors (6)
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