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Neuronal Signaling

产品 1 到 50 共 86个

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  1. Gabazine
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    Gabazine

    Catalog No. A12627
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    GABAA receptor antagonist
    Gabazine is a selective and competitive antagonist of GABAA receptor, with an IC50 of ~0.2 μM for GABA receptor. 了解更多
  2. SCH 50911
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    SCH 50911

    Catalog No. A21630
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    γ-Aminobutyric acid B GABA(B) receptor antagonist
    SCH 50911, (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid, a selective, orally-active and competitive γ-Aminobutyric acid B GABA(B) receptor antagonist. 了解更多
  3. Flumazenil
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    Flumazenil

    Catalog No. A10397
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    Benzodiazepine 拮抗剂
    Flumazenil是竞争性抑制GABA/苯二氮卓受体复合物上苯二氮卓识别位点的活性。Flumazenil在一些活性动物模型中是弱部分激动剂，但在人类中很少或没有激动剂活性。 了解更多
  4. (+)-Bicuculline
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    (+)-Bicuculline

    Catalog No. A12590
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    GABAA 拮抗剂
    (+)-Bicuculline是一种经典的GABAA拮抗剂。 了解更多
  5. 2-Hydroxysaclofen
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    2-Hydroxysaclofen

    Catalog No. A13696
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    GABAB receptors 拮抗剂
    2-Hydroxysaclofen对GABAB受体是一种有效的选择性拮抗剂。 了解更多
  6. Cloflubicyne
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    Cloflubicyne

    Catalog No. A13932
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    GABA 拮抗剂
    Cloflubicyne是一种有效的非竞争性GABA拮抗剂，惊厥药，实验室杀虫剂。 了解更多
  7. RO 15-3890
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    RO 15-3890

    Catalog No. A14349
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    benzodiazepine receptor 拮抗剂
    Ro 15-1788是苯二氮卓受体拮抗剂。 了解更多
  8. Picrotoxin
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    Picrotoxin

    Catalog No. A14004
    GABAA receptor 拮抗剂
    Picrotoxin是GABAA受体拮抗剂。该化合物已显示可增加下丘脑的去甲肾上腺素水平和周转率。 了解更多
  9. U-93631
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    U-93631

    Catalog No. A16336
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    GABAA receptor ligand
    U-93631是具有新颖化学结构的GABAA受体配体，IC50为100 nM，并且已显示在重组GABAA受体中诱导GABA诱导的全细胞Cl-电流快速，时间依赖性地衰减。 了解更多
  10. (-)-Securinine
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    (-)-Securinine

    Catalog No. A17102
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    GABA receptor 拮抗剂
    (-)-Securinine是一种最初从S. suffructicosa分离的生物碱。Securinine是一种特定的GABA受体拮抗剂，已发现在体内具有显着的CNS活性。 了解更多
  11. Cgp 52432
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    Cgp 52432

    Catalog No. A17140
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    GABA-A receptor 拮抗剂
    Cgp 52432是GABA-A受体拮抗剂。 了解更多
  12. CGP 36742
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    CGP 36742

    Catalog No. A18666
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    GABAB receptor antagonist
    CGP 36742 is a selective GABAB receptor antagonist that can penetrate the blood?Cbrain barrier after peripheral administration, with an IC50 of 32?μM. CGP 36742 is useful in treatment of depression. 了解更多
  13. Flupirtine maleate
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    Flupirtine maleate

    Catalog No. A10251
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    NMDA 拮抗剂
    Flupirtine maleate是Flupirine的盐形式，是一种非阿片类中枢性镇痛药，是一种选择性的神经元钾离子通道开放剂，也具有NMDA受体拮抗剂特性。 了解更多
  14. TCN 201
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    TCN 201

    Catalog No. A11947
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    NMDA Receptor 拮抗剂
    TCN 201是对NR1/NR2A相对于含NR1/NR2B的受体具有选择性的NMDA受体拮抗剂。 了解更多
  15. SDZ 220-581
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    SDZ 220-581

    Catalog No. A12426
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    NMDA receptor 拮抗剂
    SDZ 220-581是一种竞争性NMDA受体拮抗剂（pKi = 7.7）。 了解更多
  16. DNQX
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    DNQX

    Catalog No. A13882
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    NMDA receptor 拮抗剂
    DNQX是一种非N-甲基-D-天冬氨酸（非NMDA）受体复合物拮抗剂。 了解更多
  17. (-)-MK 801 maleate
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    (-)-MK 801 maleate

    Catalog No. A13435
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    NMDA receptor 拮抗剂.
    (-)-MK 801 maleate是一种有效的、选择性的、非竞争性的NMDA受体拮抗剂。它通过与NMDA相关离子通道内的一个位点结合而起作用。 了解更多
  18. SDZ 220-581 Ammonium salt
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    SDZ 220-581 Ammonium salt

    Catalog No. A15235
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    NMDA receptor 拮抗剂
    SDZ 220-581 Ammonium salt是NMDA谷氨酸受体亚型（pKi = 7.7）的有效竞争性拮抗剂。 了解更多
  19. L-701324
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    L-701324

    Catalog No. A15522
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    NMDA/glycine receptor 拮抗剂
    L-701324是一种活性且长效的抗惊厥药，对NMDA受体上的甘氨酸位点具有高亲和力和选择性。 了解更多
  20. (+)-MK 801 Maleate
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    (+)-MK 801 Maleate

    Catalog No. A12761
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    NMDA receptor 拮抗剂
    (+)-MK 801 Maleate是NMDA的有效拮抗剂，Ki值为30.5nM。 了解更多
  21. CGS19755
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    CGS19755

    Catalog No. A15791
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    NMDA 拮抗剂
    CGS 19755（顺式-4-膦酰基甲基-2-哌啶羧酸）是一种有效的立体定向抑制剂，由N-甲基-D-天冬氨酸（NMDA）诱发，但不是由KCl诱发的[3H]乙酰胆碱释放大鼠纹状体的切片。 了解更多
  22. Eliprodil
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    Eliprodil

    Catalog No. A12946
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    NMDA 拮抗剂
    Eliprodil是一种非竞争性NR2B-NMDA受体拮抗剂（IC50 = 1 uM），对含NR2A和NR2C的受体效力较低（IC50> 100 uM）。 了解更多
  23. GV-196771A
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    GV-196771A

    Catalog No. A13438
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    NMDA receptor antagonist
    GV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. 了解更多
  24. RPR104632
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    RPR104632

    Catalog No. A13385
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    NMDA receptor antagonist
    RPR104632 is a specific antagonist of NMDA receptor, with potent neuroprotective properties. 了解更多
  25. Ifenprodil tartrate
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    Ifenprodil tartrate

    Catalog No. A16583
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    NMDA receptor antagonist
    Ifenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). 了解更多
  26. Transcrocetinate disodium
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    Transcrocetinate disodium

    Catalog No. A21051
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    NMDA receptor antagonist
    Transcrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. 了解更多
  27. MDL 105519
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    MDL 105519

    Catalog No. A21192
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    NMDA receptor antagonist
    MDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. 了解更多
  28. Radiprodil
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    Radiprodil

    Catalog No. A21193
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    NMDA NR2B antagonist
    Radiprodil (RGH-896) is an orally active and selective NMDA NR2B antagonist. A potential therapeutic agent in treatment of neuropathic pain and possibly other chronic pain conditions. 了解更多
  29. NMDA-IN-1
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    NMDA-IN-1

    Catalog No. A21419
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    NMDA antagonist
    NMDA-IN-1 is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM. 了解更多
  30. 7-Chlorokynurenic acid sodium salt
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    7-Chlorokynurenic acid sodium salt

    Catalog No. A21879
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    NMDA receptor antagonist
    7-Chlorokynurenic acid sodium salt is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM). 了解更多
  31. SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581
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    SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581

    Catalog No. A21897
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    NMDA receptor antagonist
    SDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. 了解更多
  32. Rislenemdaz
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    Rislenemdaz

    Catalog No. A21907
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    NMDA receptor GluN2B antagonist
    Rislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. 了解更多
  33. Memantine hydrochloride
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    Memantine hydrochloride

    Catalog No. A11708
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    NMDA receptor 拮抗剂
    Memantine hydrochloride是nmda受体的拮抗剂，与离子通道位点结合。它还是CYP2B6和CYP2D6抑制剂，作用于重组CYP2B6和CYP2D6，Ki分别为0.51 nM和94.9 μM。它被用于治疗帕金森综合征。 了解更多
  34. Orphenadrine citrate
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    Orphenadrine citrate

    Catalog No. A11712
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    NMDA receptor 拮抗剂
    Orphenadrine柠檬酸盐是NMDA受体拮抗剂，Ki为6.0μM，还是HERG钾离子通道阻断剂。 了解更多
  35. Felbamate
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    Felbamate

    Catalog No. A11862
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    Felbamate是NMDA相关甘氨酸结合位点的拮抗剂。 了解更多
  36. MDL 29951
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    MDL 29951

    Catalog No. A13729
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    NMDA receptor 拮抗剂
    MDL-29951是在体外和体内均能激活NMDA受体的新型甘氨酸拮抗剂（Ki = 0.14 mM，[3H]甘氨酸结合）。 了解更多
  37. NVP-AAM077 Tetrasodium Hydrate (PEAQX)
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    NVP-AAM077 Tetrasodium Hydrate (PEAQX)

    Catalog No. A14071
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    NMDA receptors 拮抗剂
    NVP-AAM077抑制成年小鼠在脑室下区域和齿状回中的祖细胞增殖，并降低了齿状回中的新生细胞的存活。 了解更多
  38. ARL-15896
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    ARL-15896

    Catalog No. A13858
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    NMDA receptor ion channel 拮抗剂
    ARL-15896是新型的N-甲基-D-天冬氨酸受体离子通道拮抗剂。 了解更多
  39. CNQX
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    CNQX

    Catalog No. A16109
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    AMPA/kainate 拮抗剂
    CNQX是一种竞争性的非NMDA谷氨酸受体拮抗剂（AMPA和海藻酸酯受体的IC50分别为0.3和1.5 uM，而NMDA受体的IC50 = 25 uM）。 了解更多
  40. 7CKA
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    7CKA

    Catalog No. A17070
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    NMDA receptor 拮抗剂
    7CKA是在甘氨酸位点起作用的NMDA受体拮抗剂。 了解更多
  41. D-AP5
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    D-AP5

    Catalog No. A17044
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    NMDA 拮抗剂
    D-AP5是一种选择性的N-甲基-D-天冬氨酸（NMDA）受体拮抗剂，可竞争性抑制NMDA受体的谷氨酸结合位点。 了解更多
  42. Neu-2000
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    Neu-2000

    Catalog No. A17033
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    NMDA receptor 拮抗剂
    Neu-2000是可能用于治疗中风的NMDA受体拮抗剂。 了解更多
  43. Mephenesin
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    Mephenesin

    Catalog No. A17493
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    NMDA receptor antagonist
    Mephenesin is an NMDA receptor antagonist, is a centrally acting muscle relaxant. 了解更多
  44. Glycine
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    Glycine

    Catalog No. A17936
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    NMDA antagonist
    AZD-4282, also known as aminoacetic acid and glycine, is a N-methyl-D-aspartate (NMDA) receptor antagonist potentially for the treatment of neuropathic pain. 了解更多
  45. Phenoxybenzamine hydrochloride
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    Phenoxybenzamine hydrochloride

    Catalog No. A10719
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    α-adrenergic (AR) 拮抗剂/CaM 抑制剂
    Phenoxybenzamine hydrochloride是一种细胞可渗透的，非特异性的，不可逆的α-肾上腺素（AR）拮抗剂，也可作为CaM抑制剂。 了解更多
  46. Fesoterodine fumarate (Toviaz)
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    Fesoterodine fumarate (Toviaz)

    Catalog No. A10386
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    AChR 拮抗剂
    Fesoterodine fumarate是一种用于尿急的药物，可减少尿液通过的频率并促使尿失禁。 了解更多
  47. 5-hydroxymethyl tolterodine (PNU 200577)
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    5-hydroxymethyl tolterodine (PNU 200577)

    Catalog No. A11166
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    muscarinic receptor 拮抗剂
    5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物，tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。 了解更多
  48. Rocuronium bromide
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    Rocuronium bromide

    Catalog No. A10803
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    AchR 拮抗剂
    Rocuronium Bromide是一种竞争性AchR拮抗剂，用于现代麻醉中。 了解更多
  49. Biperiden HCl
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    Biperiden HCl

    Catalog No. A10147
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    Muscarinic receptor antagonist
    Biperiden HCl是毒蕈碱受体拮抗剂，对M1亚型表现出一定的选择性。 了解更多
  50. Tolterodine tartrate (Detrol LA)
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    Tolterodine tartrate (Detrol LA)

    Catalog No. A10937
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    muscarinic receptor 拮抗剂
    Tolterodine tartrate (Detrol LA)是毒蕈碱受体拮抗剂。 了解更多

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