Nexturastat A
目录号: A14032
HDAC6 抑制剂
Nexturastat A 是一种芳基脲衍生物,作为组蛋白去乙酰化酶6(HDAC6)的强效和高度选择性抑制剂(IC50= 5.02 +/- 0.60 nM)。
Discription | Nexturastat A is an aryl urea derivative that acts as a potent and highly selective inhibitor of histone deacetylase 6 (HDAC6) (IC50= 5.02 +/- 0.60 nM). | |||||
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Cell Research |
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目录号 | A14032 |
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分子式 | C19H23N3O3 |
分子量 | 341.40422 |
CAS号 | 1403783-31-2 |
SMILES | CCCCN(CC1=CC=C(C=C1)C(=O)NO)C(=O)NC2=CC=CC=C2 |
其他名称 | Nexturastat-A,NexturastatA |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 59 mg/mL (172.81 mM) | |
Water | Insoluble | ||
Ethanol | 2 mg/mL (5.85 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 29.29 mL | 146.45 mL | 292.91 mL |
0.5 mM | 5.86 mL | 29.29 mL | 58.58 mL |
1 mM | 2.93 mL | 14.65 mL | 29.29 mL |
5 mM | 0.59 mL | 2.93 mL | 5.86 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2