Octreotide Acetate
Octreotide 是一种针对 sst2、sst3 和 sst5 生长抑素受体的肽类激动剂。在克隆的人类生长抑素受体上的 IC50/Kd 值(纳摩尔)分别为:290 - 1140(sst1),0.4 - 2.1(sst2),4.4 - 34.5(sst3),> 1000(sst4),以及 5.6 - 32(sst5)。
Discription | Octreotide is a peptide agonist for sst2, sst3 and sst5 somatostatin receptors. IC50/Kd values (nM) at cloned human somatostatin receptors are: 290 - 1140 (sst1), 0.4 - 2.1 (sst2), 4.4 - 34.5 (sst3), > 1000 (sst4), and 5.6 - 32 (sst5). |
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目录号 | A12782 |
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分子式 | C49H66N10O10S2 . xC2H4O2 |
分子量 | 1019.24 (free acid) |
CAS号 | 79517-01-4 |
SMILES | CC(C1C(=O)NC(CSSCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N1)CCCCN)CC2=CNC3=CC=CC=C32)CC4=CC=CC=C4)NC(=O)C(CC5=CC=CC=C5)N)C(=O)NC(CO)C(C)O)O.CC(=O)O |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2