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Opiorphin

目录号: A23064
Opiorphin,一种阿片肽,是一种强效的人体锌外肽酶抑制剂,用于抑制脑啡肽失活。Opiorphin 抑制两种脑啡肽分解的外部酶,即人类中性外部-内部肽酶,hNEP (EC 3.4.24.11),其 IC50 值为 11 μM,以及人类外部氨基肽酶,hAP-N (EC 3.4.11.2)。Opiorphin 通过激活内源性阿片类物质依赖的传输,显示出强大的镇痛活性
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规格 价格 库存 数量
10mg
¥315.00
现货
25mg
¥665.00
现货
50mg
¥1,085.00
现货
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生物活性
Discription Opiorphin, an opioid peptide, is a potent enkephalin-inactivating zinc ectopeptidases in human inhibitor. Opiorphin inhibits two enkephalin-catabolizing ectoenzymes, human neutral ecto-endopeptidase, hNEP (EC 3.4.24.11) with an IC50 value of 11 μM, and human ecto-aminopeptidase, hAP-N (EC 3.4.11.2). Opiorphin displays potent analgesic activity by activating endogenous opioid-dependent transmission.
产品信息
目录号 A23064
分子式 C29H48N12O8
分子量 692.77
CAS号 864084-88-8
Sequence shortening QRFSR
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