PD 151746
目录号: A14245
Calpain 抑制剂
PD 151746 是一种选择性的、细胞渗透性 calpain 抑制剂,对 μ-Calpain 的 Ki 值为 0.26 uM,对 m-calpain 的选择性约为 20 倍。
Discription | PD 151746 is a selective, cell-permeable calpain inhibitor with Ki of 0.26 uM for μ-Calpain, about 20-fold selectivity over m-calpain. | ||
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Targets |
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目录号 | A14245 |
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分子式 | C11H8FNO2S |
分子量 | 237.25 |
CAS号 | 179461-52-0 |
SMILES | C1=CC2=C(C=C1F)C(=CN2)/C=C(/C(=O)O)\S |
其他名称 | PD-151746,PD151746 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 40 mg/mL (168.6 mM) | |
Water | Insoluble | ||
Ethanol | 40 mg/mL (168.6 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 42.15 mL | 210.75 mL | 421.5 mL |
0.5 mM | 8.43 mL | 42.15 mL | 84.3 mL |
1 mM | 4.21 mL | 21.07 mL | 42.15 mL |
5 mM | 0.84 mL | 4.21 mL | 8.43 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2