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PD176252

PD176252

Name: PD176252
SKU: A19385

目录号: A19385

BB1/BB2 antagonist

PD176252 Chemical Structure

CAS NO. 204067-01-6

PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; PD176252 is also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC50s of 0.31 and 0.66 μM in HL-60 cells.

库存：现货

规格	价格	数量
2 mg	￥ 840.00
5 mg	￥ 1,400.00
10 mg	￥ 2,520.00

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制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	17.1 mL	85.52 mL	171.04 mL
0.5 mM	3.42 mL	17.1 mL	34.21 mL
1 mM	1.71 mL	8.55 mL	17.1 mL
5 mM	0.34 mL	1.71 mL	3.42 mL

*The above data is based on the productmolecular weight 584.67. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A19385
作用机制	Antagonist (拮抗剂)
M. Wt	584.67
Formula	C32H36N6O5
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	204067-01-6
Synonyms	PD 176252, PD-176252
SMILES	O=C(NC1=CC=C([N+]([O-])=O)C=C1)N[C@](CC2=CNC3=C2C=CC=C3)(C)C(NCC4(C5=CC=C(OC)C=N5)CCCCC4)=O